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Antidiabetic Properties of the Histamine H3 Receptor Protean Agonist ProxyfanHENRY, Melanie B; SHUQIN ZHENG; CHENXIA DUAN et al.Endocrinology (Philadelphia). 2011, Vol 152, Num 3, pp 828-835, issn 0013-7227, 8 p.Article

Correlation of apparent affinity values from H₃-receptor binding assays with apparent affinity (pK_app) and intrinsic activity (α) from functional bioassaysHARPER, E. A; SHANKLEY, N. P; BLACK, J. W et al.British journal of pharmacology. 2007, Vol 151, Num 1, pp 128-143, issn 0007-1188, 16 p.Article

Procognitive Properties of Drugs with Single and Multitargeting H₃ Receptor Antagonist ActivitiesNIKOLIC, Katarina; FILIPIC, Slavica; AGBABA, Danica et al.CNS neuroscience & therapeutics (Print). 2014, Vol 20, Num 7, pp 613-623, issn 1755-5930, 11 p.Conference Paper

The intradermal effects of the H₃ receptor agonist R α methylhistamine in human skinKAVANAGH, G. M; SABROE, R. A; GREAVES, M. W et al.British journal of dermatology (1951). 1998, Vol 138, Num 4, pp 622-626, issn 0007-0963Conference Paper

Human skin mast cells express H2 and H4, but not H3 receptorsLIPPERT, Undine; ARTUC, Metin; KRÜGER-KRASAGAKIS, Sabine et al.Journal of investigative dermatology. 2004, Vol 123, Num 1, pp 116-123, issn 0022-202X, 8 p.Article

The histamine H3 receptor as a herapeutic drug target for CNS disoraersGEMKOW, Mark J; DAVENPORT, Adam J; HARICH, Silke et al.Drug discovery today. 2009, Vol 14, Num 9-10, pp 509-515, issn 1359-6446, 7 p.Article

Antiobesity effects of A-331440, a novel non-imidazole histamine H₃ receptor antagonistHANCOCK, Arthur A; BENNANI, Youssef L; JIA BAO PAN et al.European journal of pharmacology. 2004, Vol 487, Num 1-3, pp 183-197, issn 0014-2999, 15 p.Article

Histamine H₃-receptor agonists and imidazole-based H₃-receptor antagonists can be thermodynamically discriminatedHARPER, E. A; BLACK, J. W.British journal of pharmacology. 2007, Vol 151, Num 4, pp 504-517, issn 0007-1188, 14 p.Article

In vitro optimization of structure activity relationships of analogues of A-331440 combining radioligand receptor binding assays and micronucleus assays of potential antiobesity histamine H₃ receptor antagonistsHANCOCK, Arthur A; DIEHL, Marilyn S; COWART, Marion D et al.Basic & clinical pharmacology & toxicology (Print). 2004, Vol 95, Num 3, pp 144-152, issn 1742-7835, 9 p.Article

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New potent histamine H₃-receptor antagonists of the amide typeSTARK, H; LIPP, R; ARRANG, J.-M et al.European journal of pharmaceutical sciences. 1995, Vol 3, Num 2, pp 95-104, issn 0928-0987Conference Paper

Histamine H₃ receptor antagonists reach out for the clinicCELANIRE, Sylvain; WIJTMANS, Maikel; TALAGA, Patrice et al.Drug discovery today. 2005, Vol 10, Num 23-24, pp 1613-1627, issn 1359-6446, 15 p.Article

Alternative splicing of the histamine H₃ receptor mRNA at the third cytoplasmic loop is not detectable in humansLIU, Changlu; MA, Xiao-Jun; LOVENBERG, Timothy W et al.Molecular brain research. 2000, Vol 83, Num 1-2, pp 145-150, issn 0169-328XArticle

Subclasses of histamine H₃ antagonist binding sites in rat brainCUMMING, P; GJEDDE, A.Brain research. 1994, Vol 641, Num 2, pp 203-207, issn 0006-8993Article

Enhanced Histaminergic Neurotransmission and Steep-Wake Alterations, a Study in Histamine H3-Receptor Knock-Out MiceGONDARD, Elise; ANACLET, Christelle; AKAOKA, Hideo et al.Neuropsychopharmacology (New York, NY). 2013, Vol 38, Num 6, pp 1015-1031, issn 0893-133X, 17 p.Article

Activation of peripheral and spinal histamine H₃ receptors inhibits formalin-induced inflammation and nociception, respectivelyCANNON, Keri E; LEURS, Rob; HOUGH, Lindsay B et al.Pharmacology, biochemistry and behavior. 2007, Vol 88, Num 1, pp 122-129, issn 0091-3057, 8 p.Article

Chromosomal mapping and organization of the human histamine H₃ receptor geneTARDIVEL-LACOMBE, Joël; MORISSET, Séverine; GBAHOU, Florence et al.Neuroreport (Oxford). 2001, Vol 12, Num 2, pp 321-324, issn 0959-4965Article

Evaluation of the receptor selectivity of the H₃ receptor antagonists, iodophenpropit and thioperamide : an interaction with the 5-HT₃ receptor revealedLEURS, R; TULP, M. T. M; MENGE, M. B. P et al.British journal of pharmacology. 1995, Vol 116, Num 4, pp 2315-2321, issn 0007-1188Article

Possible participation of histamine H₃-receptors in the regulation of anaphylactic histamine release from isolated rat peritoneal mast cellsKOHNO, S; NAKAO, S; OGAWA, K et al.Japanese journal of pharmacology. 1994, Vol 66, Num 2, pp 173-180, issn 0021-5198Article

4,5-Dihydropyridazin-3-one derivatives as histamine H₃ receptor inverse agonistsHUDKINS, Robert L; AIMONE, Lisa D; ZULLI, Allison L et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 1, pp 194-198, issn 0960-894X, 5 p.Article

Localization and function of histamine H₃ receptor in the nasal mucosaSUZUKI, S; TAKEUCHI, K; MAJIMA, Y et al.Clinical and experimental allergy (Print). 2008, Vol 38, Num 9, pp 1476-1482, issn 0954-7894, 7 p.Article

Activation of histamine H₃ receptors in human nasal mucosa inhibits sympathetic vasoconstrictionVARTY, Loriann M; GUSTAFSON, Eric; LAVERTY, Maureen et al.European journal of pharmacology. 2004, Vol 484, Num 1, pp 83-89, issn 0014-2999, 7 p.Article

A qualitative model for the histamine H₃ receptor explaining agonistic and antagonistic activity simultaneouslyDE ESCH, I. J. P; TIMMERMAN, H; MENGE, W. M. P. B et al.Archiv der Pharmazie (Weinheim). 2000, Vol 333, Num 8, pp 254-260, issn 0365-6233Article

Does histamine stimulate cyclic amp formation in the avian pineal gland via a novel (non-H₁, non-H₃) histamine receptor subtypeNOWAK, J. Z; SEK, B; D'SOUZA, T et al.Neurochemistry international. 1995, Vol 27, Num 6, pp 519-526, issn 0197-0186Article